thiazol相关论文
Synthesis,fluorescence properties and selective Cr(Ⅲ) recognition of tetraaryl imidazole derivatives
Three tetraaryl imidazole derivatives 5a-5c bearing thiazole groups were synthesized in the presence of [Bmin]Br by one-......
Formation of thiazol-2(3H)-imines by reaction of α-amino acids, aroylisothiocyanates, and α-bromoket
An efficient one-pot synthesis of functionalized thiazol-2(3H)-imines by a three-component reaction between aroylisothio......
Synthesis, Crystal Structure and Fungicidal Activity of N-(4-tert-buty)-5-(1,2,4-triazol-1-yl)thiazo
The title compound has been synthesized by the reaction of 4-tert-butyl-5-(1,2,4-triazol-1-yl)-2-aminothiazole with prop......
Mannich Base Derivatives of 1,2-Benzisothiazolin-3-one: Syntheses, Crystal Structures and Bioactivit
Twelve Mannich base derivatives of 1,2-benzisothiazolin-3-one were synthesized by the reaction of 1,2-benzisothiazol-3(2......
Isoquinoline-mediated 5-vinylation and N-vinylation of benzo[d]oxazole-2-thiol and benzo[d]thiazole-
An effective route to 5-vinylated and N-vinylated benzo[d]oxazole-2(3H)-thiones and benzo[d]thiazole-2(3H)-thiones is de......
Twenty-five derivatives of glycyrrhetinic acid(GA) modified on the A-ring,at C30 and C11 positions were synthesized.Thei......
A novel and convenient synthesis of thiazolo[3,2-a]pyrimidin-7-ones and pyrido[1,2-a]pyrimidin-2-one
A novel route for the synthesis of thiazolo[3,2-a]pyrimidin-7-ones and pyrido[1,2-a]pyrimidin-2-ones from acetylated 2am......
2-(Hydrazinecarbothioyl)-N-substituted hydrazinecarbothioamides react with 2,3,5,6-tetrachloro-l,4-benzoquinone in high ......
Synthesis, Crystal Structure and DNA Interaction Study of 3-(2-(3,5-Diphenyl-4,5-dihydropyrazol-1-yl
A new compound 3-(2-(3,5-diphenyl-4,5-dihydropyrazol-1-yl)thiazol-4-yl)-2Hchromen-2-one was synthesized by cyclocondensa......
Enantioselective synthesis of β-amino esters bearing a quinazoline moiety via a Mannich-type reactio
The cinchona alkaloids catalyzed the direct asymmetric Mannich reactions of 1,3-dicarbonyl compounds with acyl imines to......
4-(7-Methoxy-2,2-dimethyl-2,3-dihydrobenzo-furan-5-yl)-N-(pyridin-2-yl)thiazol-2-amine: Chiral Cryst
The title compound 4-(7-methoxy-2,2-dimethyl-2,3-dihydrobenzofuran-5-yl)-N- (pyridin-2-yl) thiazol-2-amine was synthesiz......
Synthesis of N-substituted-2-aminobenzothiazoles using nano copper oxide as a recyclable catalyst un
A simple and practical method for the synthesis of N-substituted-2-aminobenzothiazoles via a crosscoupling reaction of 2......
A series of naphthyridinone derivatives based on la(a precursor of Voreloxin) were designed and synthesized.Seven compou......
Investigation of anticancer potencies of newly generated Schiff base imidazolylphenylheterocyclic-2-
A new series of multi-heterocyclic Schiff base was constructed starting from 4’-(imidazol-1-yl[56_TD$IF])-acetophenone ......
Antiproliferative effect of octreotide on gastric cancer cells mediated by inhibition of Akt/PKB and
AIM:To investigate the antiproliferative effect of octreotide,a long-acting analogue of somatostatin,on gastric cancerc......
Brain is very susceptible to hypo-glucose and hypoxia induced by ischemia/reperfusion and significant neuronal injuries ......
头孢菌素类抗生素发展迅速。自从分离出头孢菌素 C,改换了其母核(7-氨基头孢烷酸)第3位和第7位侧链,发展出了抗菌力强和抗菌谱广......
To study the effect of tumor necrosis factor-related apoptosis inducing ligand (TRAIL) on PC-3M cell line, PC-3M cell li......
Objective To optimize experimental parameters for the photosensitization of 5-aminolevulinic acid (ALA) in promyelocytic......
Novel ferrocenyl-containing thiazole derivatives have been synthesized from 2-amino-4-ferrocenyl-5-(1H-1, 2, 4-triazole-......
Synthesis and characterization of organotitanium substituted heteropolytungstosilicates and their bi
Tris-, di-(organotitanium) substituted tungstosilicates α、β-[(CpTi)3(SiW9O37)]7- and γ-[(Cp-Ti)2(SiW10O38)]6- were ......
The potassium dithiocarbazate 2 was obtained through condensation of 5-pyrazolehydrazide 1 with carbon disulfide in etha......
Synthesis,Crystal Structure and Antitumor Activity of Mixed Ligand Coordination Compound of Copper w
The mixed ligand coordination compound of copper with norfloxacin (NFLX) and 1, 10-phen has been synthesized and charact......
Synthesis of Novel 1-Arylsulfonyl-4-(1′-N-2′, 3′, 4′, 6′-tetra- O-acetyl-β-D-glucopyranosyl)thiosemi
The synthesis of novel 1-arylsulfonyl -4- (1′-N -2′, 3′, 4′, 6′-tetra-O-acetyl-β-D-gluco-pyranosyl) thiosemicarbaz......
Objective: A series of 2-benzylideneaminonaphthothiazoles were designed and synthesized incorporating the lipo- philic n......
Synthesis,Crystal Structure and Fungicidal Activity of(E)-2-[(4-tert-Butyl-5-(4-methoxybenzyl)thiazo
The title compound(E)-2-(4-tert-butyl-5-(4-methoxybenzyl)thiazol-2-ylimino)me-thylphenol was synthesized by the reaction......
Two novel fluorescent calix[4]arene derivatives 1a and 1b with benzoxazole or benzothiazole units in 1,3-alternate confo......
AIM:To construct the recombinant lentivirus expression plasmid,pLenti6/V5-NT4 p53(N15)-antennapedia(Ant),and study its e......
AIM:To investigate the mechanism by which galangin,a polyphenolic compound derived from medicinal herbs,induces apoptosi......
AIM:To observe the effects of sargentgloryvine stem extracts (SSE) on the hepatoma cell line HepG-2 in vitro andin vivo ......
Honokiol:a promising small molecular weight natural agent for the growth inhibition of oral squamous
Honokiol (HNK) is a small organic molecule purified from magnolia species and has demonstrated anticancer activities in ......
AIM:To observe the synergistic effects of hyperthermia in oxaliplatin-induced cytotoxicity in human colon adenocarcinoma......
AIM:To investigate the inhibitory role of toxicarioside A on the gastric cancer cell line human gastric cancer cell line......
AIM:To investigate the effect of high mobility group A2(HMGA2) gene silencing on gastric cancer MKN-45 cells in vitro.ME......
Aim: To study whether T33, a new synthesized non-thiazolidinedione (TZD) peroxisome proliferator-activated receptor (PPA......
以2-氨基-5-巯基-1，3，4-噻二唑为原料，经氯代频呐酮取代，溴代：硫脲环合得到中间体，再与一系列芳香醛和亚膦酸酯反应合成了7种目标化合物，......
胰岛β细胞数量减少和功能障碍是糖尿病的根本原因,现有的治疗手段主要以维持正常血糖水平为主要目的,尚无有效恢复受损胰岛功能的......
